Overview of Histone Deacetylase Inhibitors in Haematological Malignancies

نویسندگان

  • Mark J. Bishton
  • Ricky W. Johnstone
  • Michael Dickinson
  • Simon Harrison
  • H. Miles Prince
چکیده

Histone deacetylase inhibitors (HDACi) can induce hyperacetylation of both histone and non-histone target resulting in epigenetic reprogramming and altered activity, stability and localisation of non-histone proteins to ultimately mediate diverse biological effects on cancer cells and their microenvironment. Clinical trials have demonstrated single agent HDACi to have activity in hematological malignancies, in particular T-cell lymphoma and Hodgkin lymphoma. Combination strategies with standard therapies based on pre-clinical data are being employed with significant success due to their excellent side effect profile. Correlative studies will provide valuable information on the sub-groups of patients more likely to respond or be resistant to HDACi therapy, while long-term monitoring for toxicities is also needed.

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عنوان ژورنال:

دوره 3  شماره 

صفحات  -

تاریخ انتشار 2010